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항목
AntibodyCurated CoreFDAApproved
risankizumab-rzaa (Skyrizi, BI 655066, risankizumab)
AbbVie·IL-23 p19
110 trials·t½ 28 h
Overview
Program
Skyrizi (risankizumab-rzaa)
Overview
Company
AbbVie
Overview
Modality
ANTIBODY
Overview
Target
IL-23 p19
Overview
Indication
Plaque psoriasis, PsA, Crohn's disease, ulcerative colitis
Overview
Phase
APPROVED
Overview
Status
APPROVED
Overview
Content status
Curated Core
Overview
Data Confidence
Data Confidence · High
Overview
Development Signal
Development Signal · Established
Overview
Approval status
FDA approved
Positioning
Key differentiator
Novel therapeutic avenues, including TYK2 and HDAC inhibitors, as well as nanotechnology-based delivery systems, show encoura
Positioning
Known limitation
IL-17 independent disease and immunogenicity.
MoA
Mechanism
Risankizumab selectively binds IL-23 p19 subunit, blocking IL-23 interaction with IL-23R and downstream Th17 pathway (IL-17A/F, IL-22).
MoA
Biomarker
PASI, sPGA, IBD endoscopic scores.
PK/PD
Half-life
28 h
PK/PD
Species
Mouse
PK/PD
Animal (cat.)
Mouse
PK/PD
Experiment
Pharmacokinetic
Toxicology
Species
Cynomolgus monkey, Mouse
Toxicology
Major finding
Upper respiratory infections, headache, fatigue; low TB reactivation vs TNF class.
Toxicology
CRS
N/A
Clinical
Safety signal
Upper respiratory infections, headache, fatigue; low TB reactivation vs TNF class.
Clinical
Program phase
APPROVED
Clinical
Trial activity
No active/completed counts
Preclinical
Animal (cat.)
Mouse