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항목
AntibodyCurated CoreFDAApproved
lebrikizumab-lbkz (Ebglyss, LY3650150, lebrikizumab)
Eli Lilly·IL-13
108 trials·t½ 24.5 h
Overview
Program
Ebglyss (lebrikizumab-lbkz)
Overview
Company
Eli Lilly
Overview
Modality
ANTIBODY
Overview
Target
IL-13
Overview
Indication
Moderate-to-severe atopic dermatitis
Overview
Phase
APPROVED
Overview
Status
APPROVED
Overview
Content status
Curated Core
Overview
Data Confidence
Data Confidence · High
Overview
Development Signal
Development Signal · Established
Overview
Approval status
FDA approved
Positioning
Key differentiator
unique disposition of simvastatin rather than enzyme or transporter inhibition
Positioning
Known limitation
Concurrent IL-4 signaling and non-Type 2 dermatitis.
MoA
Mechanism
Lebrikizumab binds IL-13 with high affinity, blocking IL-13Rα1/IL-4Rα signaling and downstream Type 2 inflammation in skin (barrier dysfunction, pruritus, eosinophilia).
MoA
Biomarker
EASI, IGA 0/1, pruritus NRS.
PK/PD
Half-life
24.5 h
PK/PD
Species
NHP
PK/PD
Animal (cat.)
NHP
PK/PD
Experiment
pd
Toxicology
Species
Cynomolgus monkey, NHP
Toxicology
Major finding
Conjunctivitis, nasopharyngitis, injection-site reactions; herpes zoster warnings per class.
Toxicology
CRS
N/A
Clinical
Safety signal
Conjunctivitis, nasopharyngitis, injection-site reactions; herpes zoster warnings per class.
Clinical
Selected reported efficacy
1%
Clinical
Result source
ClinicalTrials.gov NCT03689855
Clinical
Program phase
APPROVED
Clinical
Trial activity
No active/completed counts
Clinical
Trial ref
NCT03689855
Preclinical
Animal (cat.)
Mouse