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API CSV31행 · 4개 프로그램

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항목
AntibodyCurated CoreFDAApproved
bimekizumab (Bimzelx, UCB4940, bimekizumab-bkzx)
UCB·IL-17A / IL-17F
58 trials·t½ ~23 days
AntibodyLimited DatastalePreclinical
Secikinumab (Secikinumab)
Novartis Pharmaceuticals·Psoriasis
2 trials
AntibodyCurated CorestaleApproved
Ixekizumab (Ixekizumab)
Eli Lilly and Company·Psoriatic Arthritis
53 trials·t½ 13 h
AntibodyLimited DatastalePhase 3
secukinumab (AIN457, AIN457 (secukinumab))
Novartis·Psoriatic Arthritis
148 trials·t½ 31 h
Overview
Program
Bimzelx (bimekizumab)SecikinumabIxekizumabAIN457 (secukinumab)
Overview
Company
UCBNovartis PharmaceuticalsEli Lilly and CompanyNovartis
Overview
Modality
ANTIBODYANTIBODYANTIBODYANTIBODY
Overview
Target
IL-17A / IL-17FPsoriasisPsoriatic ArthritisPsoriatic Arthritis
Overview
Indication
Plaque psoriasis, psoriatic arthritis, axial spondyloarthritis, hidradenitis suppurativaAxial Spondylarthritis (axSpA); SecukinumabPsoriasis; Atopic DermatitisAsthma
Overview
Phase
APPROVEDPRECLINICALAPPROVEDPHASE_3
Overview
Status
APPROVEDACTIVERECRUITINGACTIVE
Overview
Content status
Curated CoreLimited DataCurated CoreLimited Data
Overview
Data Confidence
Data Confidence · HighData Confidence · LowData Confidence · HighData Confidence · Low
Overview
Development Signal
Development Signal · EstablishedDevelopment Signal · WatchDevelopment Signal · EstablishedDevelopment Signal · Emerging
Overview
Approval status
FDA approvedInvestigationalApproved (flag incomplete)Investigational
Positioning
Key differentiator
IL-17F contributes independently to tissue inflammation, so blocking it as well raises the ceiling on complete skin clearance.Novel approaches, including tolerogenic DC therapy and neuroimmune modulation, hold promise for refining treatment and addres
Positioning
Known limitation
Anti-drug antibodies and non-IL-17-driven inflammatory phenotypes.
Positioning
Development positioning
Efficacy leader in psoriasis clearance versus IL-17A-only and IL-23 agents.
MoA
Mechanism
Binds IL-17A and IL-17F, preventing engagement of the IL-17RA/RC complex and shutting down downstream keratinocyte and synovial inflammatory signaling more completely than IL-17A blockade alone.targets and signaling pathwayTargeted immunotherapies provide effective interventions by disrupting these cytokine-driven pathway
MoA
Biomarker
PASI/IGA response, hs-CRP in axial disease.biomarkers and optimize therapeutic strategies
PK/PD
Half-life
~23 days13 h31 h
PK/PD
Species
Cynomolgus monkey, PASI 90/100, HiSCR in HS, ASAS40 in axSpAMouseRat, Human
PK/PD
Animal (cat.)
Human, NHP, In vitroMouseHuman, Rat
PK/PD
Experiment
pdpharmacokineticPD
Toxicology
Species
Cynomolgus monkeyMouseRat, Human
Toxicology
Animal (cat.)
MouseHuman, Rat
Toxicology
Major finding
Oral candidiasis is the signature toxicity of IL-17F co-blockade and occurs in roughly 10–20% of patients. Upper respiratory infection is common; inflammatory bowel disease requires monitoring.Ixekizumab Treatment Persistence in Psoriatic Arthritis: Response to Joaquin et al.. We appreciate the interest of Joaquin et al in our recent study on the treatment persistence of ixekizumab in psoriatic arthritis. In response, we clarify that our study utilized prospectively collected real-world clinical data from a multicenter observational cohort, rather than administrative databases. We empha…Effectiveness of brodalumab in biologic-experienced adults with moderate to severe plaque psoriasis: a focused narrative review.. To summarize recent literature evaluating treatment outcomes in adults with plaque psoriasis who switched to brodalumab from a different biologic because of treatment failure (inadequate initial response/loss of an adequate initial response) and/or adverse events. Relev…
Toxicology
CRS
N/A
Clinical
Safety signal
Oral candidiasis is the signature toxicity of IL-17F co-blockade and occurs in roughly 10–20% of patients. Upper respiratory infection is common; inflammatory bowel disease requires monitoring.Ixekizumab Treatment Persistence in Psoriatic Arthritis: Response to Joaquin et al.. We appreciate the interest of Joaquin et al in our recent study on the treatment persistence of ixekizumab in psoriatic arthritis. In response, we clarify that our study utilized prospectively collected real-world clinical data from a multicenter observational cohort, rather than administrative databases. We empha…Effectiveness of brodalumab in biologic-experienced adults with moderate to severe plaque psoriasis: a focused narrative review.. To summarize recent literature evaluating treatment outcomes in adults with plaque psoriasis who switched to brodalumab from a different biologic because of treatment failure (inadequate initial response/loss of an adequate initial response) and/or adverse events. Relev…
Clinical
Selected reported efficacy
9%
Clinical
PASI75
PASI 100 than secukinumab at week 16 and mai
Clinical
Result source
BE RADIANT (NCT03536884) / BE VIVID / BE SUREClinicalTrials.gov NCT03131570
Clinical
Program phase
APPROVEDPRECLINICALAPPROVEDPHASE_3
Clinical
Trial activity
No active/completed countsNo active/completed counts
Clinical
Trial ref
NCT03536884NCT03131570