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항목
AntibodyCurated CoreFDAApproved
atezolizumab (Tecentriq, MPDL3280A)
Roche / Genentech·PD-L1
693 trials·t½ 27 h
Overview
Program
Tecentriq (atezolizumab)
Overview
Company
Roche / Genentech
Overview
Modality
ANTIBODY
Overview
Target
PD-L1
Overview
Indication
NSCLC, SCLC, HCC, TNBC, urothelial carcinoma, and others
Overview
Phase
APPROVED
Overview
Status
APPROVED
Overview
Content status
Curated Core
Overview
Data Confidence
Data Confidence · High
Overview
Development Signal
Development Signal · Established
Overview
Approval status
FDA approved
Positioning
Key differentiator
novel agents have been approved in recent years (including systemic pembrolizumab, nogapendekin alfa inbakicept-pmln, N-803),
Positioning
Known limitation
resistance to existing therapies
MoA
Mechanism
Atezolizumab binds PD-L1 and blocks its interaction with PD-1 and B7.1 (CD80), enabling restoration of antitumor T-cell responses without direct PD-1 engagement on T cells.
MoA
Biomarker
PD-L1 IC/TC scoring in NSCLC and UC; tumor-type-specific thresholds.
PK/PD
Half-life
27 h
PK/PD
Species
Mouse, Human
PK/PD
Animal (cat.)
Human, Mouse
PK/PD
Experiment
PD
Toxicology
Species
Cynomolgus monkey, Mouse, Human
Toxicology
Major finding
Immune-mediated pneumonitis, hepatitis, colitis, endocrinopathies.
Toxicology
CRS
N/A
Clinical
Safety signal
Immune-mediated pneumonitis, hepatitis, colitis, endocrinopathies.
Clinical
Reported PFS
1.7
Clinical
Reported OS
7.6
Clinical
Result source
ClinicalTrials.gov NCT04457778
Clinical
Program phase
APPROVED
Clinical
Trial activity
No active/completed counts
Clinical
Trial ref
NCT04457778
Preclinical
Animal (cat.)
Mouse