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검색으로 10,000+ 프로그램 중 최대 5개를 골라 PK/PD · 독성 · 임상을 나란히 비교합니다. · 다음 갱신 D-8 · 마지막 7월 21일

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API CSV23행 · 1개 프로그램

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항목
ADCPreclinical
Targeted drugs (Targeted drugs)
Ascendis Pharma Endocrinology Divi…·Immune-related Adverse Event
ORR 15%
Overview
Program
Targeted drugs
Overview
Company
Ascendis Pharma Endocrinology Division A/S
Overview
Modality
ADC
Overview
Target
Immune-related Adverse Event
Overview
Indication
Immune-related Adverse Event; Malignant Solid Tumors
Overview
Phase
PRECLINICAL
Overview
Status
RECRUITING
MoA
Mechanism
target-mediated or intrinsic, which requires only the intrinsic half-life and the target receptor
MoA
Biomarker
biomarker-guided precision strategy integrated with modern systemic therapy
PK/PD
Species
Rat
PK/PD
Animal (cat.)
Rat, In vitro
PK/PD
Experiment
PK
Toxicology
Species
Rat
Toxicology
Animal (cat.)
Rat, In vitro
Toxicology
Major finding
Comprehensive Evaluation of YJ-2 as a PAD4 Inhibitor in Alleviating Ischemic Brain Injury: From NETs-Induced Neurotoxicity to In Vivo Neuroprotection.. To evaluate the neuroprotective potential of YJ-2, a novel peptidylarginine deiminase 4 (PAD4) inhibitor, against ischemia/reperfusion brain injury by targeting neutrophil extracellular trap (NET) formation. In vitro, a NETs-induced injury mod…
Clinical
Primary efficacy
ORR 15%
Clinical
ORR
15%
Clinical
PFS
59.1
Clinical
OS
59.1
Clinical
Result source
ClinicalTrials.gov NCT02285439
Clinical
Data Tier / Score
A · 38
Clinical
Program phase
PRECLINICAL
Clinical
Clinical sync
2026년 7월 18일 (8일 전)